Naphthyridine integrase inhibitors
Filed: May 12th, 2004 [Pending]
Patent Application Number: 10556311
N(R4)C(0)0R4, — N(R4)C(R4)(0), - — NS(0)2NR4, — R3N(R4)S(0)2R4, — R3S(0)2NR4 -N( R4)R3N(R4)2 — N(R4)C(0)R4, — N(R4)C(0)C(0)N(R4)2, — N(R4)C(R4)(0), ...
4-AMINO-2,3-DISUBSTITUTED THIENO [2,3,D]PYRIMIDINES AND PHARMACEUTICAL ...
Filed: July 9th, 2008 [Pending]
Patent Application Number: 12169800
... heteroaryl, aryl or heteroaryl substituted with at least one independently selected R group, heterocyclyl, — RR3, — C(0)0R4, — C(0)NR5R6, or — C(0)R4; ...
Compounds for the treatment of inflammatory disorders
Filed: January 16th, 2007 [Pending]
Patent Application Number: 11653798
... the group consisting of a covalent bond, -(C(R4)2)n-, -N(R4)-, -^(O)N(R4) ... N(R4)— S(0)2— , — O— , — S— , — C(O)— , — S(O)— , and — S(0)2— ; m is 1 to ...
IMIDAZO[5,1-C][1,2,4]BENZOTRIAZINE DERIVATIVES AS INHIBITORS OF ...
Filed: November 6th, 2009 [Pending]
Patent Application Number: 12614146
R4, halo, cyano, nitro, — NR5R6, — C(0)NR5R6, — S(0)2— NR5R6, — N(R7)— C (O)— NR8R9, — N(R10)— C(O)— R4, and — N(R10)— C(O) O — R4; wherein said alkyl, ...
Benzimidazoles
Filed: January 4th, 2005 [Pending]
Patent Application Number: 11029064
... cyano, halo, haloalkyl, hydroxy, nitro, R4, — C(=0)R4, — C(=0)NY1Y2, — C(=0) 0R4, — N(R6)C(=0)R4, — N(R6)C(=0)NY1Y2, — N(R6)C(=0)OR4, — N(R6)S02R4, ...
Piperidinyl targeting compounds that selectively bind integrins
Filed: February 18th, 2004 [Pending]
Patent Application Number: 10782060
... Rj is — N(R4)(R6), -heterocyclyl(R8) or -heteroaryl(R8); Rla is -C(R4)(=N-R4 ), _C(=N-R4)-N(R4)2, _C(=N-R4)-N(R4)(R6), _C(=N-R4)- N(R4)— C(=0)— R4, ...
Compounds and methods for the treatment of cardiovascular, inflammatory and ...
Filed: October 9th, 1996 [Granted]
Patent Number: 6420392
5 10 wherein: Ar1 is either 15 20 25 and wherein: W is independently selected from the group consisting of: 35 — AN(OM)C(0)N(R3)R4, — AN(R3)C(0)N(OM)R4, ...
SPIRO (FURO [3, 2-C] PYRIDINE-3-3' -INDOL) -2' (1'H)-ONE DERIVATIVES AND ...
Filed: October 12th, 2007 [Pending]
Patent Application Number: 12445270
... R9 — OC(O) R5, — R9— C(0)OR5, — R9— C(0)N(R4)R5, — R9— C(0)R5, — R9— OR5 or— R9— CN; R12 is hydrogen, alkyl, aryl, aralkyl or — C(0)R5 ...