X1 X2 R1 R5a 1-46 FF Pn 4PP-NH 5 1-126 CI H Me cPn-NH 1-47 FF Hx ECM-NH 1-127 CI H Me 2.4DFP-NH 1-48 FF Me 1AD-NH 1-49 FF Me 3.5DFP-NH 1-50 FF Me 2-Pym-NH ...

The amount of reagent to be used in the reaction is usually 1 mole of the ... B 1-1 F CI H CH3 HH 1-2 F CI H CH3 H OH 1-3 F CI H CH3 H OCH3 1-4 F CI H CH3 ...

... H 98 TABLE 6a-continued (If-a) NaW B OCH3 CI H OCH3 CI H 25 OCH3 CI H A. ... C3H7 H CI H 6-OCH3 i-C3H7 H CI H 6-OCH3 C4H9 H CI H 6-OCH3 i-C4H9 H CI H ...

Y R' R a MX n Yield (%) 1 CHj HH 2 Zn CI 2 92 2 CH3 HH 2 Zn SO4 1 71 3 CH3 HH 1 Cu CI 2 47 4 CH3 CI H 2 Zn CI 2 95 5 CH3 CI H 2 Zn Br 2 80 6 CH3 CI H 2 Zn 1 ...

XY R3 R1 R2 B 1-529 H CI H CF3 CH3 S'C3H7 1-530 H CI H CF3 CH3 SCH2CH2C1 1-531 H CI H CF3 CH3 S C5Hg 1-532 H CI H CF3 CH3 SCC6H11 1-533 H CI H CF3 CH3 ...

... 1 2 C(=0)CH3 CH2Br F CN CHC1 1 2 C02CH3 CH2C1 F CN CHC1 1 2 C02CH3 CH2Br F CN CHC1 1 2 CH2C=CH CH2C1 F CN CHC1 1 2 CH2C=CH CH2Br CI H CH2 1 1 H CH2C1 CI ...

88 TABLE 1 '-continued 139a 1 — CH, ON CI CI H 140a 1 — CH.CH, ON CI CI H 141a 1 HON CI CI H 142a 1 — CH, ON CI CI H 143a 0 HON CI CI H 144a 1 — CH, ...

HC(=S)CF3 CF3 CI H CF3 H CI 379. H CF3 CI CI H CF3 H CI 380. H CF3 CN CI H CF3 H CI 381. H SCCI2F H CI H CI H OCH3 382. H SOCCl2F H CI H CI H OCH3 383.