Substituted 1,2,4-triazole angiotensin II antagonists
Filed: March 8th, 1991 [Granted]
Patent Number: 5093346
Rl R2 R3 R5 A mp (°C.) 235 n-propyl CH2SO2CH3 C02H H Single bond 236 n-propyl CH =CHCH2OH C02H H Single bond 237 n-propyl CH=CHCH2OCH3 C02H H Single bond 238 ...
Substituted pyrazole angiotensin II antagonists
Filed: August 5th, 1992 [Granted]
Patent Number: 5315013
R' R2 R3 R5 A 113 n-propyl O || C02H H Single bond CH2SCH3 o 114 n-propyl CH= CHCH2OH C02H H Single bond 115 n-propyl CH=CHCH2OCH3 C02H H Single bond 116 ...
Substituted 1,2,3 triazole angiotensin II antagonists
Filed: July 10th, 1991 [Granted]
Patent Number: 5189048
235 n-propyl CH2S02CH3 C02H H Single bond 236 n-propyl CH=CHCH2OH C02H H Single bond 237 n-propyl CH=CHCH2OCH3 C02H H Single bond 238 n-propyl CH=CHCH2OEt ...
Substituted pyrrole angiotensin II antagonists
Filed: March 26th, 1990 [Granted]
Patent Number: 5043349
55 56 TABLE 2-continued 1,2,4-TRIAZOLES N — NN R3 R5 A C02H H Single C02H ... 113 n-propyl O || C02H H Single bond CH2SCH3 O 114 n-propyl CH=CHCH2OH C02H H ...
Treatment of hypertension with 1,2,4-angiotensin II antagonists
Filed: December 6th, 1988 [Granted]
Patent Number: 5015651
65 66 TABLE 3-continued PYRAZOLES R2 NR? R3 ^ C02H N— Ph mp CO ... CH2SCH3 235 n -propyl CH2SO2CH3 C02H H Single bond 236 n-propyl CH=CHCH2OH C02H H Single ...
Sulphamides for Treatment of Cancer
Filed: May 16th, 2006 [Pending]
Patent Application Number: 11920450
[0103] In further examples of embodiment (A), R2 is H, R14 is n-propyl, ... —CHO , — C02H, — CH=CHC02Me, — CH=CHC02H, — CH=CHCH2OH, — CH=N— OH, — CH=N— OEt, ...
Treatment of congestive heart failure with angiotensin 11 receptor blocking ...
Filed: November 13th, 1989 [Granted]
Patent Number: 5128355
=„,o coy 314 1 n-butyl CI CH=CHCH2OH C02H ^> N = N / \ N NH ... 312 1 n-propyl H CH2OH C02H 313 1 n-pentyl CI CH2OH 103-104.5 314A 1 n-butyl CF3 ...
Sulfamides as gamma-secretase inhibitors
Filed: October 29th, 2001 [Granted]
Patent Number: 7138400
... R2 is H, R14 is n-propyl, and R4 is — CH=CHCH2N(R16)2 where 5 — N(Ri6)2 is ... C02H, — CH=CHC02Me, — CH=CHC02H, — CH=CHCH2OH, — CH=N— OH, — CH=N— OEt, ...